NA-Semax Amidate

N-Acetyl Semax Amidate · NASA

Rank#999
CognitiveNot ApprovedApprovedResearchIntranasal

Popular for:Enhanced cognitive version of Semax, longer-acting, BDNF stimulation

0

Total Studies

0

Human Studies

Approved

Evidence Level

Not Approved

FDA Status

Overview

NA-Semax Amidate (N-Acetyl Semax Amidate) is a modified version of the Russian nootropic peptide Semax, with two chemical modifications: an N-terminal acetyl group and a C-terminal amide group. These modifications increase the peptide's stability, bioavailability, and duration of action compared to standard Semax.

The acetylation protects against aminopeptidase degradation while the amidation protects against carboxypeptidase degradation, effectively shielding both ends of the peptide from enzymatic breakdown. This results in a longer-acting and more potent version that has become the preferred form in the Western research peptide community.

Mechanism of Action

Like standard Semax, NA-Semax Amidate is a synthetic analog of ACTH (4-10) that stimulates BDNF (Brain-Derived Neurotrophic Factor) and NGF (Nerve Growth Factor) expression. It modulates serotonergic, dopaminergic, and cholinergic neurotransmitter systems. The enhanced stability from the acetyl and amide modifications means higher effective concentrations reach target neural tissues, potentially producing stronger neurotrophic effects per dose compared to standard Semax.

Key Research Benefits

Enhanced stability and potency vs standard Semax
Stimulates BDNF and NGF expression
Studied for cognitive enhancement and neuroprotection
Longer duration of action (less frequent dosing)
Modulates multiple neurotransmitter systems simultaneously

Clinical Evidence Summary

Research Pipeline

Preclinical
Animal
Phase I
Phase II
Phase III
Approved

International Regulatory Status

🇷🇺
RussiaApproved1996(Semax (parent compound))

Cognitive disorders (approved as parent compound Semax)

Source

0

Total Studies

0

Human Studies

Not FDA-approved. Modified version of Russian-approved Semax. Research compound. Popular in nootropics community as the preferred Semax variant.

Key Studies / PubMed References

Therapeutic Peptides in Orthopaedics: Applications, Challenges, and Future Directions.

Review

Rahman OF, Lee SJ, Seeds WA · Journal of the American Academy of Orthopaedic Surgeons. Global research & reviews · 2026

PMID: 41490200

Semax peptide targets the μ opioid receptor gene Oprm1 to promote deubiquitination and functional recovery after spinal cord injury in female mice.

Animal Study

Liu R, Chen Y, Huang H, et al. · British journal of pharmacology · 2025

PMID: 40692165

ACTH-like Peptides Compensate Rat Brain Gene Expression Profile Disrupted by Ischemia a Day After Experimental Stroke.

Animal Study

Filippenkov IB, Shpetko YY, Stavchansky VV, et al. · Biomedicines · 2024

PMID: 39767736

[The efficacy of semax in the tretament of patients at different stages of ischemic stroke].

Human Study

Gusev EI, Martynov MY, Kostenko EV, et al. · Zhurnal nevrologii i psikhiatrii imeni S.S. Korsakova · 2018

PMID: 29798983

Pharmacological Aspects of Neuro-Immune Interactions.

Review

Tarasov VV, Kudryashov NV, Chubarev VN, et al. · Current pharmaceutical design · 2018

PMID: 28875850

Side Effects & Safety

Nasal irritation
Headache (usually resolves after first few days)
Mild anxiety in sensitive individuals (due to stimulating nature)
Insomnia if dosed too late in the day

Known Interactions

No curated interaction entry is live for NA-Semax Amidate yet.

Until the interaction table is fully populated, use the interaction checker and related peptides below to explore adjacent compounds and likely research pairings.

Frequently Asked Questions

Research Disclaimer

This page is for research and educational purposes only. The information presented is based on published scientific literature and does not constitute medical advice, diagnosis, or treatment recommendations. NA-Semax Amidate is not approved by the FDA for human therapeutic use. Always consult a qualified healthcare professional before making any health-related decisions. The studies referenced are linked to their original PubMed sources for verification.