Epithalon

Epitalon · Epithalamin · AEDG

Anti-AgingNot ApprovedApprovedResearchSubQ

Popular for:Telomerase activation, anti-aging, pineal gland function

0

Registered Trials

7

Trial Publications

189

PubMed References

Approved

Evidence Level

Overview

Epithalon (also spelled Epitalon) is a synthetic tetrapeptide (Ala-Glu-Asp-Gly) studied for its effects on telomerase activation and potential anti-aging properties. The short version: people usually care about it for telomerase activation, anti-aging, pineal gland function, but the strength of the evidence depends heavily on indication and study type.

Epithalon (also spelled Epitalon) is a synthetic tetrapeptide (Ala-Glu-Asp-Gly) studied for its effects on telomerase activation and potential anti-aging properties. It is based on the naturally occurring pineal gland peptide Epithalamin, researched extensively by Russian gerontologist Professor Vladimir Khavinson over several decades.

Khavinson's research suggests that Epithalon may activate telomerase, the enzyme responsible for maintaining telomere length, which is a key biomarker of cellular aging. His studies, primarily conducted in Russia, report effects on lifespan extension in animal models and melatonin normalization.

Research Snapshot

What the evidence says

Approved

Epithalon currently shows 0 registered trials from ClinicalTrials.gov, 7 PubMed trial publications (5 RCT-tagged), and 189 PubMed references matching the stored source query. Treat PubMed references as literature surface area, not a count of clinical trials.

Known vs uncertain

Known signals

  • 0 registered trials are tracked from ClinicalTrials.gov intervention records.
  • 7 PubMed clinical-trial publications are indexed.
  • 5 PubMed randomized controlled trial publications are indexed.
  • 189 PubMed references are tracked separately from trial counts and can include animal, in-vitro, review, mechanism, or clinical records.

Open questions

  • Evidence strength may vary by indication, route, formulation, and population.
  • Public anecdotes can highlight interest or concern but do not establish clinical efficacy.
  • Regulatory status and compounding access can change independently from the research literature.

Mechanism of Action

Epithalon is studied for its ability to activate telomerase reverse transcriptase (hTERT), the catalytic subunit of telomerase.

Key Research Benefits

Studied for telomerase activation and telomere maintenance
Researched for pineal gland function and melatonin normalization
Khavinson studies report lifespan extension in animal models
May support circadian rhythm regulation
Studied for retinal health and degenerative conditions

Clinical Evidence Summary

Research Pipeline

Preclinical
Animal
Phase I
Phase II
Phase III
Approved

International Regulatory Status

🇷🇺
RussiaApproved2001(Epithalamin)

Geroprotective (anti-aging), immune modulation

Source

0

Registered Trials

7

Trial Publications

5

RCT Publications

189

PubMed References

ClinicalTrials.govPubMed ESearchCurated alias queryChecked May 3, 2026

Registered trials are ClinicalTrials.gov intervention records. Trial publications are PubMed records tagged as clinical trials or randomized controlled trials. PubMed references are broader source-query matches and can include animal studies, in-vitro work, reviews, mechanism papers, and trial publications.

0

Registered trials

7

Trial publications

5

RCT publications

189

PubMed references

19

Reviews

0

Meta-analyses

Registered trials source

Jun 1, 2026

Epithalon

Uses the exact compound name as a ClinicalTrials.gov intervention query.

View source

Publication counts source

May 3, 2026

Epithalon, Epitalon, Epithalamin, AEDG

Uses common transliterations and product names for this peptide family.

View source

Not FDA-approved. Primarily studied in Russian academic research (Khavinson, St. Petersburg Institute of Bioregulation and Gerontology). Limited Western clinical trial data. Research compound.

Key PubMed References

189 PubMed references · showing top 25 by relevance

View all on PubMed

Therapeutic Peptides in Orthopaedics: Applications, Challenges, and Future Directions.

Review

Rahman OF, Lee SJ, Seeds WA · Journal of the American Academy of Orthopaedic Surgeons. Global research & reviews · 2026

PMID: 41490200

Epitalon increases telomere length in human cell lines through telomerase upregulation or ALT activity.

In Vitro

Al-Dulaimi S, Thomas R, Matta S, et al. · Biogerontology · 2025

PMID: 40908429

Overview of Epitalon-Highly Bioactive Pineal Tetrapeptide with Promising Properties.

Review

Araj SK, Brzezik J, Mądra-Gackowska K, et al. · International journal of molecular sciences · 2025

PMID: 40141333

The Antioxidant Tetrapeptide Epitalon Enhances Delayed Wound Healing in an in Vitro Model of Diabetic Retinopathy.

In Vitro

Gatta M, Dovizio M, Milillo C, et al. · Stem cell reviews and reports · 2025

PMID: 40493162

Peptide Regulation of Cell Differentiation.

In Vitro

Khavinson V, Linkova N, Diatlova A, et al. · Stem cell reviews and reports · 2020

PMID: 31808038

Anecdotes & Sentiment

Public discussion, not clinical evidence

This section summarizes what people are talking about in public sources. It can be useful for spotting questions, hype cycles, and recurring concerns, but it is separate from the evidence sections above.

No curated public-discussion themes are live for Epithalon yet.

Side Effects & Safety

- Generally well-tolerated in available research - Injection site reactions - Limited human safety data from Western clinical trials - Long-term effects not fully characterized

Generally well-tolerated in available research
Injection site reactions
Limited human safety data from Western clinical trials
Long-term effects not fully characterized

Known Interactions

No curated interaction entry is live for Epithalon yet.

Until the interaction table is fully populated, use the interaction checker and related peptides below to explore adjacent compounds and likely research pairings.

Comparison Pages

Comparison pages

All

No comparison page is linked yet.

Frequently Asked Questions

Research Disclaimer

This page is for research and educational purposes only. The information presented is based on published scientific literature and does not constitute medical advice, diagnosis, or treatment recommendations. Regulatory status can vary by compound, formulation, indication, and jurisdiction. Check official labeling, registry records, and qualified professional guidance before making any health-related decision. The studies referenced are linked to their original PubMed sources for verification.