Thymosin Alpha-1

Ta1 · Zadaxin · Thymalfasin

ImmuneNot ApprovedApprovedMixedSubQ

Popular for:Immune modulation, T-cell function, hepatitis treatment

61

Registered Trials

49

Trial Publications

575

PubMed References

Approved

Evidence Level

Overview

Thymosin Alpha-1 (Ta1) is a 28-amino acid peptide naturally produced by the thymus gland that plays a crucial role in immune system regulation. The short version: people usually care about it for immune modulation, t-cell function, hepatitis treatment, but the strength of the evidence depends heavily on indication and study type.

Thymosin Alpha-1 (Ta1) is a 28-amino acid peptide naturally produced by the thymus gland that plays a crucial role in immune system regulation. It is approved as a pharmaceutical drug (Zadaxin) in over 30 countries for the treatment of hepatitis B, hepatitis C, and as an immune adjuvant.

Thymosin Alpha-1 is one of the most clinically validated peptides, with extensive human trial data. The thymus gland shrinks with age (thymic involution), and declining Ta1 levels are associated with age-related immune dysfunction. Exogenous Ta1 supplementation is studied for restoring T-cell function and immune surveillance.

Research Snapshot

What the evidence says

Approved

Thymosin Alpha-1 currently shows 61 registered trials from ClinicalTrials.gov, 49 PubMed trial publications (35 RCT-tagged), and 575 PubMed references matching the stored source query. Treat PubMed references as literature surface area, not a count of clinical trials.

Known vs uncertain

Known signals

  • 61 registered trials are tracked from ClinicalTrials.gov intervention records.
  • 49 PubMed clinical-trial publications are indexed.
  • 35 PubMed randomized controlled trial publications are indexed.
  • 575 PubMed references are tracked separately from trial counts and can include animal, in-vitro, review, mechanism, or clinical records.

Open questions

  • Evidence strength may vary by indication, route, formulation, and population.
  • Public anecdotes can highlight interest or concern but do not establish clinical efficacy.
  • Regulatory status and compounding access can change independently from the research literature.

Mechanism of Action

Thymosin Alpha-1 enhances T-cell maturation, differentiation, and function by acting on toll-like receptors (TLR2, TLR9) in dendritic cells.

Key Research Benefits

Approved as Zadaxin in 30+ countries for hepatitis B/C
Enhances T-cell maturation and function
Studied for immune reconstitution in aging and immunodeficiency
Researched as vaccine adjuvant (improves vaccine efficacy)
Investigated for cancer immunotherapy support
One of the most clinically validated peptides

Clinical Evidence Summary

Research Pipeline

Preclinical
Animal
Phase I
Phase II
Phase III
Approved

International Regulatory Status

🇨🇳
ChinaApproved1996(Zadaxin)

Hepatitis B, hepatitis C, immune deficiency, adjunct cancer therapy

Source

61

Registered Trials

49

Trial Publications

35

RCT Publications

575

PubMed References

ClinicalTrials.govPubMed ESearchExact-name queryChecked May 3, 2026

Registered trials are ClinicalTrials.gov intervention records. Trial publications are PubMed records tagged as clinical trials or randomized controlled trials. PubMed references are broader source-query matches and can include animal studies, in-vitro work, reviews, mechanism papers, and trial publications.

61

Registered trials

49

Trial publications

35

RCT publications

575

PubMed references

76

Reviews

10

Meta-analyses

Registered trials source

Jun 1, 2026

Thymosin Alpha-1

Uses the exact compound name as a ClinicalTrials.gov intervention query.

View source

Publication counts source

May 3, 2026

Thymosin Alpha-1

Uses the exact display name.

View source

Approved as Zadaxin in 30+ countries (not FDA-approved in US). Extensive human clinical trial data. FDA Category 2 status under review; potential Category 1 reinstatement.

Key PubMed References

575 PubMed references · showing top 25 by relevance

View all on PubMed

The efficacy and safety of thymosin alpha-1 combined with lenvatinib plus sintilimab in unresectable hepatocellular carcinoma: a retrospective study.

Human Study

Yao S, Huang Q, Zou Y, et al. · Scientific reports · 2025

PMID: 40263352

Aging and Thymosin Alpha-1.

Review

Simonova MA, Ivanov I, Shoshina NS, et al. · International journal of molecular sciences · 2025

PMID: 41373628

Phenotypic drug discovery: a case for thymosin alpha-1.

Review

Garaci E, Paci M, Matteucci C, et al. · Frontiers in medicine · 2024

PMID: 38903817

Enhanced Immunomodulatory Effects of Thymosin-Alpha-1 in Combination with Polyanionic Carbosilane Dendrimers against HCMV Infection.

In Vitro

Espinar-Buitrago MS, Magro-López E, Vázquez-Alejo E, et al. · International journal of molecular sciences · 2024

PMID: 38396631

Comprehensive Review of the Safety and Efficacy of Thymosin Alpha 1 in Human Clinical Trials.

Review

Dinetz E, Lee E · Alternative therapies in health and medicine · 2024

PMID: 38308608

Anecdotes & Sentiment

Public discussion, not clinical evidence

This section summarizes what people are talking about in public sources. It can be useful for spotting questions, hype cycles, and recurring concerns, but it is separate from the evidence sections above.

No curated public-discussion themes are live for Thymosin Alpha-1 yet.

Side Effects & Safety

- Generally very well-tolerated in clinical trials - Injection site reactions - Rare cases of mild fever (immune activation) - Fatigue during initial use

Generally very well-tolerated in clinical trials
Injection site reactions
Rare cases of mild fever (immune activation)
Fatigue during initial use

Known Interactions

No curated interaction entry is live for Thymosin Alpha-1 yet.

Until the interaction table is fully populated, use the interaction checker and related peptides below to explore adjacent compounds and likely research pairings.

Comparison Pages

Comparison pages

All

No comparison page is linked yet.

Frequently Asked Questions

Research Disclaimer

This page is for research and educational purposes only. The information presented is based on published scientific literature and does not constitute medical advice, diagnosis, or treatment recommendations. Regulatory status can vary by compound, formulation, indication, and jurisdiction. Check official labeling, registry records, and qualified professional guidance before making any health-related decision. The studies referenced are linked to their original PubMed sources for verification.